Vesicle-based formulations for pain treatment: a narrative review. [Review]

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All Authors

Martinez, J.
Ingram, N.
Kapur, N.
Jayne, DG.
Beales, PA.

LTHT Author

Jayne, David

LTHT Department

General Surgery

Non Medic

Publication Date

2024

Item Type

Journal Article
Review

Language

Subject

Subject Headings

Abstract

Pain, a complex and debilitating condition, necessitates innovative therapeutic strategies to alleviate suffering and enhance patients' quality of life. Vesicular systems hold the potential to enhance precision of drug localisation and release, prolong the duration of therapeutic action and mitigate adverse events associated with long-term pharmacotherapy. This review critically assesses the current state-of-the-art in vesicle-based formulations (liposomes, polymersomes, ethosomes, and niosomes) for pain management applications. We highlight formulation engineering strategies used to optimise drug pharmacokinetics, present preclinical findings of experimental delivery systems, and discuss the clinical evidence for the benefits of clinically approved formulations. We present the challenges and outlook for future improvements in long-acting anaesthetic and analgesic formulation development.

Journal

The Pain Report